| Description |
FDA Indication |
Alkeran®
(Melphalan)
Alkylating agents, Nitrogen mustards |
Ovarian cancer, multiple myeloma |
Arimidex®
(Anastrozole)
Hormones, Aromatase inhibitors |
Breast cancer |
Aromasin®
(Exemestane)
Hormones, Aromatase inhibitors |
Breast cancer |
Casodex™
(Bicalutamide)
Hormones, Antiandrogens |
Prostate cancer |
CeeNU®
(Lomustine)
Alkylating agents, Nitrosoureas |
Brain tumors, Hodgkin's lymphoma |
Cytoxan®
(Cyclophosphamide)
Alkylating agents, Nitrogen mustards |
non-Hodgkin's lymphoma and Hodgkin's lymphoma, leukemia, breast cancer, multiple myeloma, Neuroblastoma, Retinoblastoma, Mycosis Fungoides (cutaneous T-cell lymphoma), ovarian cancer |
Emcyt®
(Estramustine)
Alkylating agents, Estrogen/Nitrogen mustards |
Prostate cancer |
Ergamisol®
(Levamisole)
Biological response modifiers |
Colorectal cancer |
Eulexin®
(Flutamide)
Hormones, Antiandrogens |
Prostate cancer |
Fareston®
(Toremifene)
Hormones, Antiestrogens |
Breast cancer |
Femara®
(Letrozole)
Hormones, Aromatase inhibitors |
Breast cancer |
Gleevec®
(Imatinib)
Protein-Tyrosine Kinase inhibitors |
Chronic myeloid leukemia (CML), gastrointestinal stromal tumors (GIST) |
Hexalen®
(Altretamine)
Alkylating agents, ethylenimines/methylamines |
Ovarian cancer |
Hydrea®
(Hydroxyurea)
Substituted ureas |
Melanoma; resistant chronic myelocytic leukemia; recurrent, metastatic, or inoperable carcinoma of the ovary. Head and neck cancer |
Leukeran®
(Chlorambucil)
Alkylating agents, Nitrogen mustards |
Chronic lymphatic (lymphocytic) leukemia (CLL), malignant lymphomas including lymphosarcoma, giant follicular lymphoma and Hodgkin's lymphoma |
Lysodren®
(Mitotane)
Miscellaneous |
Adrenal cortical carcinoma |
Matulane®
(Procarbazine)
Mehtylhydrazine |
Hodgkin's lymphoma |
Megestrol(Generic)
Hormone Progestine |
Breast or Endometrial Cancer |
Myleran®
(Busulfan)
Alkylating agents, Alkyl sulfonates |
Chronic myelogenous (myeloid, myelocytic, granulocytic) leukemia (CML) |
Nexavar®
(Sorafenib) |
Kidney cancer |
Nilandron®
(Nilutamide)
Hormones, Antiandrogens |
Prostate cancer |
Purinethol®
(Mercaptopurine)
Antimetabolites, Purine analogs |
Acute lymphatic (lymphocytic, lymphoblastic) leukemia, Acute myelogenouse (and acute myelomonocytic) leukemia |
Revlimid®
(Lenalidomide)
Immunomodulators |
Multiple myeloma.
Transfusion-dependent anemia due to low-or-intermediate-1-risk myelodysplastic syndromes. |
Soltamox®
(Tamoxifen Citrate)
Hormones, Antiestrogens |
breast cancer |
Sprycel™
(Dasatinib) |
chronic, accelerated, or myeloid or lymphoid blast phase chronic myeloid leukemia (CML) with resistance or intolerance to prior therapy including imatinib. Dasatinib is also FDA approved for the treatment of adults with Philadelphia chromosone-positive acute lymphoblastic leukemia (Ph+ ALL) |
Sutent®
(Sunitinib)
Multikinase inhibitor |
Kidney cancer |
Tabloid®
(Thioguanine)
Antimetabolites, Purine analogs |
Acute nonlymphocytic leukemias |
Tamoxifen
Hormones, Antiestrogens |
Breast cancer |
Tarceva®
(Erlotinib)
Epidermal Growth Factor Receptor Inhibitors |
non-small cell lung cancer and pancreatic cancer |
Targretin®
(Bexarotene)
Retinoids |
Cutaneous manifestations of cutaneous T-cell lymphoma (CTCL) |
Temodar®
(Temozolomide)
Imidazotetrazine |
Anaplastic astrocytoma, glioblastoma multiforme |
Teslac®
(Testolactone)
Hormones, Androgens |
Breast cancer |
Thalomid®
(Thalidomide)
Antiangiogenetic Agents |
Multiple myeloma
Treatment and maintenance therapy for prevention and suppresion of Erythema Nosoum Leprosum |
Trexall™
(Methotrexate)
Alkylating Agents, Folic Acid Antagonists |
Breast cancer, head and neck, advanced mycosis fungoides (cutaneous T-cell lymphoma) and lung cancer, particularly squamous cell and small cell types; in combination therapy in the treatment of advanced-stage non-Hodgkin's lynphomas (NHL) |
VePesid®
(Etoposide)
Epipodophyllotoxins, Podophyllotoxins |
Small cell lung cancer |
Vesanoid®
(Tretinoin)
Retinoids |
Acute promyelocytic leukemia |
Xeloda®
(Capecitabine)
Antimetabolites, Pyrimidine analogs |
Colorectal cancer, breast cancer |